Which is better for melasma tranexamic acid or azelaic acid?

Author: Yolanda O'Reilly  |  Last update: Monday, June 9, 2025

One small study did reveal that a combination of oral and topical 3% tranexamic acid had a significantly better outcome than a combination of oral tranexamic acid and 20% azelaic acid. ¹⁰ This might suggest a stronger impact of TXA on melasma, but it's important to remember that research in this area is still limited.

Which acid is best for melasma?

Background: Melasma is a common acquired disorder of hyperpigmentation that commonly affects those with skin of color. Tranexamic acid (TXA) is a novel treatment for melasma that has a multimodal mechanism of action.

Can azelaic acid get rid of melasma?

Azelaic acid works by inhibiting melanin pigment production. This helps to reduce the amount of pigment that is produced in areas affected by melasma. Also, azelaic acid promotes cell turnover and exfoliates the skin, which can help remove the excess pigmented cells contributing to melasma.

What is the fastest treatment for melasma?

Triple combination cream for melasma

Dr. Fernandez says that one of the best treatment cream for melasma is a triple-combination cream consisting of hydroquinone, tretinoin, and a topical corticosteroid. What makes this medication so effective is that it addresses melasma from three different angles.

Does tranexamic acid remove melasma?

Melasma is a prevalent and challenging skin condition that affects the face and causes distress in many patients and physicians. Tranexamic acid (TA) has been found to be effective for treating melasma and can be administered through multiple routes.

Should you use Azelaic acid for Pigmentation? | Dr Davin Lim

Which is better for hyperpigmentation tranexamic acid or azelaic acid?

Are you confused about whether tranexamic acid or azelaic acid is better for dark spots and discoloration? Ultimately, choosing the best of these two acids comes down to personal preference and skin tolerance, because both are relatively gentle options that offer exceptional support for minimizing hyperpigmentation.

What is the best remover for melasma?

The most commonly used treatments for melasma are skin lightening medications that are applied topically. These include medications such as hydroquinone, azelaic acid, kojic acid, niacinamide, cysteamine, rucinol, and tranexamic acid.

What is the ultimate remedy for melasma?

Retinol can reduce melasma by inhibiting the activity of melanocytes (the cells responsible for producing melanin). By modulating the skin's response to UV exposure and reducing tyrosinase enzyme activity, retinol helps reduce melasma pigmentation.

What is the 3 cream for melasma?

Tri-Luma (fluocinolone/hydroquinone/tretinoin) - Uses, Side Effects, and More. Overview: Tri-Luma is used to treat a condition called melasma, which is where colored areas appear on the face. Tri-Luma contains three medicines.

What is the best ingredient to remove melasma?

Hydroquinone is one of the most commonly prescribed treatments for melasma. It works by inhibiting the production of melanin in the skin.

Can I use tranexamic and azelaic acid together?

Can I use tranexamic acid and azelaic acid at the same time? Yes, you can generally use tranexamic acid and azelaic acid together, and there are several prescription and over-the-counter products that contain both. In fact, Curology offers personalized formulas with one or both of these proven ingredients.

What is better than azelaic acid?

If you have extremely dry skin, you may find that niacinamide is better than azelaic acid due to its ability to support the skin's natural protective barrier (and thus, encourage moisture retention).

Which is better for melasma, hydroquinone or azelaic acid?

We conclude that azelaic acid may be better than hydroquinone in reducing melasma severity as measured by the MASI. However, no significant difference between both treatments regarding the side effects.

How long does it take for tranexamic acid to work for melasma?

How long should you take oral tranexamic acid for melasma to see gains? Oral tranexamic acid treatment benefits maximize after taking it for eight to twelve weeks. During this time, it limits a cellular process involved in producing melanin, the pigment that makes your skin dark and causes freckles.

What is the new treatment for melasma?

Topical proton pump inhibitors (PPIs), such as omeprazole, may also inhibit melanogenesis, and present a promising treatment for melasma. Omeprazole topically applied onto the skin of UV-irradiated human subjects elicited significant reduction of pigment levels after 3 weeks compared to untreated controls46.

How long does it take for azelaic acid to work on melasma?

You should expect to see some improvement quite quickly - in 6 weeks or so, things should start to look better. But for clearance of pigmentation, you may well be looking at 6 months +, for issues like post-inflammatory hyperpigmentation in acne in those with melanated skin.

What actually gets rid of melasma?

The combination of hydroquinone, tretinoin and a moderate topical steroid has had the best effect on melasma. Other agents that are being studied to improve melasma include: Absorbic acid (vitamin C).

Which acid removes melasma?

In studies, tranexamic acid has been shown to decrease the patches of melasma when other treatments fail to work.

What is the new trio for melasma?

Investigators involved in a recent study 1 found that a New Trio (NT) combination cream containing isobutylamido-thiazolyl-resorcinol, retinoic acid, and dexamethazone was efficacious in the treatment of melasma and may serve as an alternative to the melasma gold-standard treatment, known as Kligman's Trio (KT).

What is the gold standard for melasma?

Hydroquinone. HQ is the most frequently prescribed depigmenting agent worldwide and it has remained the gold standard for the treatment of melasma, particularly of the epidermal type.

What cancels out melasma?

Prioritizing your skincare routine and using products containing niacinamide, vitamin C and alpha hydroxy acids are essential for helping hyperpigmentation fade over time, celebrity makeup artist, Marco Antonio says. Applying a daily SPF is recommended for preventing and diminishing the appearance of melasma.

What is the permanent cure for melasma?

Most dermatologists start Melasma treatment in India with a topical therapy. The aim of treatment of Melasma on face is to stop the melanocytes from forming any new pigments. Most commonly for the treatment of Melasma on face Hydroquinone is used.

What do Koreans use for melasma?

In conclusion, Korean red ginseng powder showed good tolerability and beneficial effects in patients with melasma. The use of Korean red ginseng would be counted as a useful adjunctive therapy for patients with melasma.

How did I cured my melasma naturally?

Aloe vera is a fantastic melasma treatment at home, known for its soothing and healing properties. Applying fresh aloe vera gel to affected areas can help reduce pigmentation and improve overall skin health. Leave the gel on for 20-30 minutes before rinsing.

What is the best vitamin to remove melasma?

What other vitamins can treat melasma?
  • Vitamin C (as antioxidants)
  • Vitamin E & fish oil (antioxidants)
  • Green tea (taste good, acts as overall antioxidant for the body & skin)

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